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BT2

Glpbio
Catalog No:GC38014-10mM (in 1mL DMSO) CAS No.:34576-94-8 MDLNo: Brand:Glpbio purity: 特性: Purpose:BT2 是 BCKDC 激酶 (BDK) 抑制剂,IC50 值为 3.19 μM。BT2 与 BDK 的结合会触发支链 α-酮酸脱氢酶复合物 (BCKDC) 的 N 末端结构域的螺旋运动,从而导致 BDK 与 BCKDC 分离。BT2 (compound 4) 也是一种有效的选择性的 Mcl-1 抑制剂,Ki 值为 59 μM。DMSO: 83.33 mg/mL (337.23 mM)
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